

HY-163065 · 50 mg
MedChemExpress · Cat: HY-163065
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medchemexpress.com/%CF%831-receptor-%CE%BC-opioid-receptor-m...Description
?1 Receptor/? Opioid receptor modulator 2 compound 4x is a dual ?OR agonist/?1R antagonist, and displays picomolar ?OR agonism activity EC50: 0.6 AAasAasAA+/- 0.2 nM and good ?1R inhibitory activity Ki: 363.7 AAasAasAA+/- 5.6 nM . ?1 Receptor/? Opioid receptor modulator 2 exhibits robust analgesic effects in various pain models.