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2?-Thioadenosine
GENERAL CATALOGUE

2?-Thioadenosine

HY-137028 · 50 mg

MedChemExpress · Cat: HY-137028

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Catalog No: HY-137028
CAS No: 136904-69-3
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress

Description

2-Thioadenosine PD157432 is a selective and irreversible inhibitor of ErbB-1 and ErbB-2, with an IC50 of 45 AAasAasAAmuM for ErbB-2. 2-Thioadenosine covalently inactivates ErbB-1 via modification of a cysteine residue at the active site.

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