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(3S)-Tanzisertib hydrochloride
GENERAL CATALOGUE

(3S)-Tanzisertib hydrochloride

HY-15495B · 50 mg

MedChemExpress · Cat: HY-15495B

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Catalog No: HY-15495B
CAS No: 2517855-91-1
Category: Apoptosis
Pack Size: 50 mg
Brand: MedChemExpress

Description

3S -Tanzisertib hydrochloride 3S -CC-930 hydrochloride is an orally active JNK inhibitor IC50 values for JNK1, JNK2, and JNK3 are 61, 7, and 6 nM, respectively . 3S -Tanzisertib hydrochloride selectively inhibits ERK1, p38?, and EGFR IC50 = 0.48, 3.4, and 0.38 ?M, respectively . 3S -Tanzisertib hydrochloride inhibits LPS-induced TNF? production in an acute rat PK-PD model. 3S -Tanzisertib hydrochloride can be used in idiopathic pulmonary fibrosis IPF research.

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