

HY-157425 · 50 mg
MedChemExpress · Cat: HY-157425
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/5-ht2cr-agonist-1.html
Description
5-HT2CR agonist 1 compound 8 , a 7-chloro analogue, is a selective 5-HT2CR partial agonist Emax=71.09 % with an EC50 value of 121.5 nM and no observed activity toward 5-HT2AR or 5-HT2BR. 5-HT2CR agonist 1 exhibits no recruitment activity for ?-arrestin and shows low inhibition of hERG at 10 ?M.







