

HY-125957 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-125957
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medchemexpress.com/a-3-hydrochloride.htmlDescription
A-3 hydrochloride is a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases. It against PKA Ki=4.3 AAasAasAAmuM , casein kinase II Ki=5.1 AAasAasAAmuM and myosin light chain kinase MLCK Ki=7.4 AAasAasAAmuM . A-3 hydrochloride also inhibits PKC and casein kinase I with Ki values of 47 AAasAasAAmuM and 80 AAasAasAAmuM, respectively.





