

HY-155245 · 1 mg
MedChemExpress · Cat: HY-155245
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Manufacturer product page
medchemexpress.com/a09-003.html
Description
A09-003 is a CDK-9 inhibitor IC50: 16 nM . A09-003 inhibits leukemia cell proliferation IC50: 1.90, 0.86, 2.49, 1.84, 0.48 ?M for BDCM, Molm-14, THP-1, U937, MV4-11 cells . A09-003 induces apoptosis and decreases Mcl-1 expression through Thr163 dephosphorylation.







