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[Ala17]-MCH TFA
GENERAL CATALOGUE

[Ala17]-MCH TFA

HY-P1204A · 50 mg

MedChemExpress · Cat: HY-P1204A

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medchemexpress.com/ala17-mch-tfa.html
Catalog No: HY-P1204A
Category: GPCR G Protein
Pack Size: 50 mg
Brand: MedChemExpress

Description

Ala17 -MCH TFA, a MCH analogue HY-P1525A , is a selective ligand for MCHR1 Ki=0.16 nM over MCHR2 Ki=34 nM . Eu3+ chelate-labeled Ala17 -MCH shows high affnity for MCHR1 Kd=0.37 nM while has little demonstrable binding affnity for MCHR2.

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