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Avatrombopag maleate
GENERAL CATALOGUE

Avatrombopag maleate

HY-13463A · Free Sample (0.1 - 0.2 mg)

MedChemExpress · Cat: HY-13463A

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Catalog No: HY-13463A
CAS No: 677007-74-8
Category: Immunology Inflammation
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress

Description

Avatrombopag AKR-501 maleate is an orally active, non-peptide thrombopoietin receptor TPO receptor agonist EC50: 3.3 nM . Avatrombopag maleate mimics the biological activity of TPO. Avatrombopag maleate increases platelet production by activating intracellular signaling systems and promotes the production of platelets and megakaryocytes from hematopoietic precursor cells. Avatrombopag maleate is a substrate for cytochrome P450 CYP 2C9 and CYP3A .

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