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Avitinib
GENERAL CATALOGUE

Avitinib

HY-19816 · Free Sample (0.1 - 0.2 mg)

MedChemExpress · Cat: HY-19816

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medchemexpress.com/avitinib.html
Catalog No: HY-19816
CAS No: 1557267-42-1
Category: Apoptosis
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress

Description

Avitinib Abivertinib is a third-generation, irreversible and orally active selective EGFR inhibitor, with IC50 values of 0.18 nM, 0.18 nM, 7.68 nM and against EGFR L858R, EGFR T790M and wild-type EGFR. Avitinib is also a BTK inhibitor that induces apoptosis and inhibits phosphorylation of BTK in mantle cell lymphoma. Avitinib shows anticancer effects.

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