

HY-170776 · 50 mg
MedChemExpress · Cat: HY-170776
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medchemexpress.com/axl-angiokinase-in-1.htmlDescription
AXL/Angiokinase-IN-1 compound 11b is an AXL/triple angiokinase inhibitor, IC50=3.75 nM AXL expression . AXL/Angiokinase-IN-1 inhibits epithelial-mesenchymal transition EMT in Bxpc-3, blocking lung cancer cell metastasis. AXL/Angiokinase-IN-1 also inhibits vascular and fibroblast functions, promoting apoptosis apoptosis in cancer cells and fibroblasts. AXL/Angiokinase-IN-1 features low toxicity and good metabolic stability.







