

HY-119682 · 50 mg
MedChemExpress · Cat: HY-119682
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medchemexpress.com/bax-agonist-1.htmlDescription
Bax agonist 1 compound SMBA2 is a Bax agonist Ki=57.2 nM . Bax agonist 1 induces Bax conformational changes by blocking S184 phosphorylation, promoting Bax insertion into the mitochondrial membrane and forming Bax oligomers, which induce cytochrome c release and apoptosis in malignant cancer cells expressing Bax. Bax agonist 1 can be used in lung cancer research.







