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BDP9066
GENERAL CATALOGUE

BDP9066

HY-111424 · Free Sample (0.1 - 0.2 mg)

MedChemExpress · Cat: HY-111424

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Catalog No: HY-111424
CAS No: 2226507-04-4
Category: Cytoskeleton
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress

Description

BDP9066 is a potent and selective myotonic dystrophy-related Cdc42-binding kinase MRCK inhibitor with an IC50 of 64 nM for MRCK? in SCC12 cells, Ki values of 0.0136 nM and 0.0233 nM for MRCK?/? in house determinations, respectively. BDP9066 has therapeutic effect on skin cancer by reducing substrate phosphorylation.

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