

HY-15150R · 5 mg
MedChemExpress · Cat: HY-15150R
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medchemexpress.com/bemcentinib-standard.htmlDescription
Bemcentinib Standard is the analytical standard of Bemcentinib. This product is intended for research and analytical applications. Bemcentinib R428 is a selective and orally active Axl inhibitor with an IC50 of 14 nM. Bemcentinib retards cancer cell migration and invasion. Bemcentinib exhibits >100-fold selectivity for Axl versus Abl and 50- and >100-fold selectivity over TAM family kinases Mer and Tyro3, respectively, in cells. Bemcentinib blocks tumor spread and prolongs survival in models of metastatic breast cancer.







