

HY-131061 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-131061
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Manufacturer product page
medchemexpress.com/bet-bromodomain-inhibitor-1.html
Description
BET bromodomain inhibitor 1 is an orally active, selective bromodomain and extra-terminal BET bromodomain inhibitor with an IC50 of 2.6 nM for BRD4. BET bromodomain inhibitor 1 binds to BRD2 2 , BRD3 2 , BRD4 1 , BRD4 2 , and BRDT 2 with high affinities Kd values of 1.3 nM, 1.0 nM, 3.0 nM, 1.6 nM, 2.1 nM, respectively . bromodomain inhibitor 1 has anti-cancer activity.

