GENERAL CATALOGUE
BI-9321
HY-114208 · 50 mg
MedChemExpress · Cat: HY-114208
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/bi-9321.htmlCatalog No: HY-114208
CAS No: 2387510-86-1
Category: Epigenetics
Pack Size: 50 mg
Brand: MedChemExpress
Description
BI-9321, a chemical probe, is a potent, selective and cellular active nuclear receptor-binding SET domain 3 NSD3 -PWWP1 domain antagonist with a Kd value of 166 nM. BI-9321 is inactive against NSD2-PWWP1 and NSD3-PWWP2. BI-9321 specifically disrupts histone interactions of the NSD3-PWWP1 domain with an IC50 of 1.2 ?M in U2OS cells.