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BMS-818251
GENERAL CATALOGUE

BMS-818251

HY-125183 · 50 mg

MedChemExpress · Cat: HY-125183

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medchemexpress.com/bms-818251.html
Catalog No: HY-125183
CAS No: 2974489-09-1
Category: Anti-infection
Pack Size: 50 mg
Brand: MedChemExpress

Description

BMS-818251 is a potent, small-molecule inhibitor of HIV-1 entry with an EC50 value of 0.019 nM. BMS-818251 shows >10-fold higher potency than BMS-626529 HY-15440 on a cross-clade panel of 208-HIV-1 strains. BMS-818251 interacts with gp120 residues from the conserved ?20-?21 hairpin to improve potency.

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