GENERAL CATALOGUE
BMY 28674
HY-100057 · 1 mg
MedChemExpress · Cat: HY-100057
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medchemexpress.com/bmy-28674.htmlCatalog No: HY-100057
CAS No: 125481-61-0
Category: GPCR G Protein
Pack Size: 1 mg
Brand: MedChemExpress
Description
BMY 28674 6-Hydroxybuspirone is the active metabolite of the anxiolytic buspirone HY-B1115A and is metabolized by CYP3A4.4. BMY 28674 binds to the serotonin 5-HT receptor subtype 5-HT1A in the rat hippocampus and dorsal raphe EC50s are 4 and 1 ?M, respectively and is an antagonist of dopamine D2, D3, and D4 receptors IC50s are 3.1, 4.9, and 0.85 ?M, respectively . BMY 28674 also inhibits organic cation transporter 1 OCT1 , OCT2, and OCT3 expressing human transporters in S2 proximal tubule cells in a concentration-dependent manner.
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