

HY-120765 · 50 mg
MedChemExpress · Cat: HY-120765
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Manufacturer product page
medchemexpress.com/brd2879.html
Description
BRD2879 is a potent IDH1-R132H inhibitor with IC50 values of 0.05, 2.5, >20, >20 AAasAasAAmuM for IDH1-R132H, IDH1-R132C, IDH1-WT, IDH2-R140Q, respectively. BRD2879 reduces R -2-hydroxyglutarate R-2HG levels.