

HY-149519 · 50 mg
MedChemExpress · Cat: HY-149519
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Manufacturer product page
medchemexpress.com/brd4-inhibitor-28.html
Description
BRD4 Inhibitor-28 Compound 18 is an orally active BRD4 Inhibitor. BRD4 Inhibitor-28 inhibits BRD40-BD1, BRD40-BD2 with IC50s of 15, 55 nM. BRD4 Inhibitor-28 also inhibits BRD2-BD1, BRD3-BD1, BRDT-BD1 with IC50s of 19, 25, 68 nM. BRD4 Inhibitor-28 has anti-melanoma activity.