

HY-156152 · 50 mg
MedChemExpress · Cat: HY-156152
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medchemexpress.com/protac-carm1-degrader-1.htmlDescription
PROTAC CARM1 degrader-1 compound 3b is a degrader DC50=8.1 nM of co-activator associated argininemethyltransferase CARM1 . PROTAC CARM1 degrader-1 degrades CARM1 in a VHL- and proteasome-dependent manner. Thus, PROTAC CARM1 degrader-1 inhibits methylation of CARM1 substrates such as poly A -binding protein PABP1 and BGR1-associated factor BAF155 and inhibits breast cancer cell migration.

