

HY-156153 · 50 mg
MedChemExpress · Cat: HY-156153
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medchemexpress.com/protac-carm1-degrader-2.htmlDescription
PROTAC CARM1 degrader-2 compound 3e is a degrader DC50=8.8 nM of co-activator associated argininemethyltransferase CARM1 . PROTAC CARM1 degrader-2 degrades CARM1 in a VHL- and proteasome-dependent manner. Thus, PROTAC CARM1 degrader-2 inhibits methylation of CARM1 substrates such as poly A -binding protein PABP1 and BGR1-associated factor BAF155 and inhibits breast cancer cell migration.

