GENERAL CATALOGUE
CCG258208
HY-109562 · 50 mg
MedChemExpress · Cat: HY-109562
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Manufacturer product page
medchemexpress.com/grk2-in-1.htmlCatalog No: HY-109562
CAS No: 2055990-90-2
Category: GPCR G Protein
Pack Size: 50 mg
Brand: MedChemExpress
Description
CCG258208 GRK2-IN-1 is a potent and selective GRK2 G protein-coupled receptor kinase 2 inhibitor IC50=30 nM while maintaining 230-fold selectivity over GRK5 IC50=7.09 ?M and more than 2500-fold selectivity over GRK1 IC50=87.3 ?M , PKA, and ROCK1. CCG258208 can be used in heart failure research.
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