

HY-109562A · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-109562A
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medchemexpress.com/grk2-in-1-hydrochloride.htmlDescription
CCG258208 GRK2-IN-1 hydrochloride is a potent and selective GRK2 G protein-coupled receptor kinase 2 inhibitor IC50=30 nM while maintaining 230-fold selectivity over GRK5 IC50=7.09 ?M and more than 2500-fold selectivity over GRK1 IC50=87.3 ?M , PKA, and ROCK1. CCG258208 hydrochloride can be used in heart failure research.







