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CDK/HDAC-IN-2
GENERAL CATALOGUE

CDK/HDAC-IN-2

HY-146276 · 50 mg

MedChemExpress · Cat: HY-146276

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Manufacturer product page

medchemexpress.com/cdk-hdac-in-2.html
Catalog No: HY-146276
CAS No: 2580938-58-3
Category: Apoptosis
Pack Size: 50 mg
Brand: MedChemExpress

Description

CDK/HDAC-IN-2 is a potent HDAC/CDK dual inhibitor with IC50 of 6.4, 0.25, 45, >1000, 8.63, 0.30, >1000 nM for HDAC1, HDAC2, HDAC3, HDAC6,8, CDK1, CDK2, CDK4,6,7, respectively. CDK/HDAC-IN-2 shows excellent antiproliferative activities. CDK/HDAC-IN-2 induces apoptosis and cell cycle arrest at G2/M phase. CDK/HDAC-IN-2 shows potent antitumor efficacy.

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