

HY-106993A · 1 mg
MedChemExpress · Cat: HY-106993A
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medchemexpress.com/cipralisant-maleate.htmlDescription
Cipralisant GT-2331 maleate is an orally active, low-toxicity, potent, selective, high affinity histamine H3 receptor full antagonist in vivo, and an agonist in vitro, with a pKi of 9.9 for histamine H3 receptor and a Ki of 0.47 nM for rat histamine H3 receptor. Cipralisant maleate has the potential for attention-deficit hyperactivity disorder research. Cipralisant maleate is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition CuAAc with molecules containing Azide groups.







