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cis-NVP-ADW742
GENERAL CATALOGUE

cis-NVP-ADW742

HY-10252A · 50 mg

MedChemExpress · Cat: HY-10252A

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Catalog No: HY-10252A
CAS No: 475489-15-7
Category: Apoptosis
Pack Size: 50 mg
Brand: MedChemExpress

Description

cis-NVP-ADW742 cis-ADW742 is a cis isomer of NVP-ADW742 HY-10252 . NVP-ADW742 is an orally active, selective IGF-1R tyrosine kinase inhibitor with an IC50 of 0.17 ?M. NVP-ADW742 inhibits insulin receptor InsR with an IC50 of 2.8 ?M. NVP-ADW742 induces pleiotropic antiproliferative/proapoptotic biologic sequelae in tumor cells.

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