

HY-17366 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-17366
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Manufacturer product page
medchemexpress.com/Clozapine-N-oxide.html
Description
Clozapine N-oxide is a major metabolite of Clozapine and a human muscarinic designer receptors DREADDs agonist. Clozapine N-oxide activates the DREADD receptor hM3Dq and hM4Di. Clozapine N-oxide cant cross the blood-brain barrier. Clozapine is a potent dopamine antagonist and also a potent and selective muscarinic M4 receptor EC50=11 nM agonist.







