

HY-103045 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-103045
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medchemexpress.com/cmpd101.htmlDescription
CMPD101 is a potent, highly selective and membrane-permeable small-molecule inhibitor of GRK2/3 with IC50 of 18 nM and 5.4 nM, respectively. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKC? with IC50s of 3.1 ?M , 2.3 ?M, 1.4 ?M and 8.1 ?M, respectively. CMPD101 can be used for the study of heart failure.