

HY-N2453 · 1 mg
MedChemExpress · Cat: HY-N2453
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medchemexpress.com/convallatoxin.htmlDescription
Convallatoxin is a cardiac glycoside isolated from Adonis amurensis Regel et Radde. Convallatoxin ameliorates colitic inflammation via activation of PPAR? and suppression of NF-?B. Convallatoxin is a P-glycoprotein P-gp substrate and recognized Val982 as an important amino acid involved in its transport. Convallatoxin is an enhancer of ligand-induced MOR endocytosis with high potency and efficacy. Anti-inflammatory and anti-proliferative properties.