

HY-P10948 · 50 mg
MedChemExpress · Cat: HY-P10948
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Manufacturer product page
medchemexpress.com/cs-vip-8.html
Description
CS-VIP 8 is a selective allosteric WDR5 protein inhibitor Ki= 0.008 ?M . CS-VIP 8 induces conformational changes in the MLL1 complex, leading to the dissociation of MLL1 from the complex, inhibiting MLL1 histone methyltransferase activity and regulating HOX gene expression. CS-VIP 8 is promising for research of hematological diseases such as leukemia.

