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CSI86
GENERAL CATALOGUE

CSI86

HY-169378 · 50 mg

MedChemExpress · Cat: HY-169378

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medchemexpress.com/csi86.html
Catalog No: HY-169378
Category: Apoptosis
Pack Size: 50 mg
Brand: MedChemExpress

Description

CSI86 is a MYC-targeting PROTAC degrader with antiproliferative activity IC50: 13-18 ?M . CSI86 is composed of MYC inhibitor red part CSI118 TFA HY-169379 , E3 ligase ligand blue part VH032 HY-120217 , and PROTAC linker black part Succinic anhydride HY-79369 . The conjugate composed of E3 ligase ligand and linker is S,R,S -CO-C2-acid HY-131866 .

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