

HY-121638 · 50 mg
MedChemExpress · Cat: HY-121638
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Manufacturer product page
medchemexpress.com/cu-3.html
Description
CU-3 is the racemate of 5Z,2E -CU-3. 5Z,2E -CU-3 is a potent and selective inhibitor against the ?-isozyme of DGK with an IC50 value of 0.6 ?M, competitively inhibits the affinity of DGK? for ATP with a Km value of 0.48 mM. 5Z,2E -CU-3 targets the catalytic region, but not the regulatory region of DGK?. 5Z,2E -CU-3 has antitumoral and proimmunogenic effects, enhances the apoptosis of cancer cells and the activation of T cells.







