

HY-146401 · 50 mg
MedChemExpress · Cat: HY-146401
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/cxcr4-antagonist-6.htmlDescription
CXCR4 antagonist 6 compound 46 is a potent CXCR4 antagonist with an IC50 value of 79 nM. CXCR4 antagonist 6 inhibits CXCL12 induced cytosolic calcium flux IC50 = 0.25 nM . CXCR4 antagonist 6 significantly mitigates CXCL12/CXCR4 mediated cell migration. CXCR4 antagonist 6 exhibits marked efficacy in a cancer metastasis model in mice.







