

HY-10968A · 50 mg
MedChemExpress · Cat: HY-10968A
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medchemexpress.com/cym5442-hydrochloride.htmlDescription
CYM5442 hydrochloride is a potent, highly-selective and orally active sphingosine 1-phosphate S1P1 receptor agonist with an EC50 of 1.35 nM. CYM5442 hydrochloride is inactive against S1P2, S1P3, S1P4, and S1P5. CYM5442 hydrochloride activates S1P1-dependent p42/p44-MAPK phosphorylation. CYM5442 exerts retinal neuroprotection. CYM5442 hydrochloride can easily penetrate the central nervous system CNS .







