

HY-10861 · 5 mg
MedChemExpress · Cat: HY-10861
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medchemexpress.com/d3-5-ht-receptor-modulator-1.htmlDescription
D3/5-HT receptor modulator-1 compound 5i is a selective dopamine D3 receptor and 5-HT2A receptor antagonist and a partial 5-HT1A receptor agonist. D3/5-HT receptor modulator-1 shows Ki values of 4.5 nM, 11.9 nM, and 15.3 nM for dopamine D3, 5-HT2A, and 5-HT2A receptors. D3/5-HT receptor modulator-1 has a low affinity for dopamine D2 receptors, 5-HT2C receptors, and hERG channels. D3/5-HT receptor modulator-1 has an atypical antipsychotic profile.