

HY-19981B · 50 mg
MedChemExpress · Cat: HY-19981B
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medchemexpress.com/derazantinib-dihydrochloride.htmlDescription
Derazantinib ARQ-087 dihydrochloride is an ATP competitive and orally activeFGFR inhibitor IC50s: 1.8 nM for FGFR2, 4.5 nM for FGFR1 and 3 . Derazantinib dihydrochloride inhibits FGFR phosphorylation. Derazantinib dihydrochloride inhibits tumor growth in multiple xenograft models.







