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Derazantinib dihydrochloride
GENERAL CATALOGUE

Derazantinib dihydrochloride

HY-19981B · 50 mg

MedChemExpress · Cat: HY-19981B

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Catalog No: HY-19981B
CAS No: 1821329-75-2
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress

Description

Derazantinib ARQ-087 dihydrochloride is an ATP competitive and orally activeFGFR inhibitor IC50s: 1.8 nM for FGFR2, 4.5 nM for FGFR1 and 3 . Derazantinib dihydrochloride inhibits FGFR phosphorylation. Derazantinib dihydrochloride inhibits tumor growth in multiple xenograft models.

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