GENERAL CATALOGUE
Didesmethyl cariprazine
HY-100658 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-100658
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medchemexpress.com/didesmethyl-cariprazine.htmlCatalog No: HY-100658
CAS No: 839712-25-3
Category: GPCR G Protein
Pack Size: 10 mM * 1 mL in DMSO
Brand: MedChemExpress
Description
Didesmethyl cariprazine is an orally active, BBB-permeable metabolite of Cariprazine HY-14763 . Didesmethyl cariprazine is a partial agonist at the D2 and D3 receptors, full agonist at the 5-HT1A receptor, and antagonist at the human 5-HT2B receptor Ki: 1.41 nM human D2L , 0.056 nM human D3 , 1.7 nM human 5-HT1A , 0.52 nM human 5-HT2B . Didesmethyl cariprazine dose-dependently inhibits the spontaneous activity of rat midbrain dopaminergic neurons.
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