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DSP-1053 benzenesulfonate
GENERAL CATALOGUE

DSP-1053 benzenesulfonate

HY-111419A · 50 mg

MedChemExpress · Cat: HY-111419A

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Catalog No: HY-111419A
CAS No: 1176326-78-5
Category: GPCR G Protein
Pack Size: 50 mg
Brand: MedChemExpress

Description

DSP-1053, a benzylpiperidine derivative, is a potent serotonin transporter SERT inhibitor with a Ki of 1.02 nM. DSP-1053 shows partial 5-HT1A receptor agonistic activity with a Ki of 5.05 nM. DSP-1053 has antidepressant activity.

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