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DXR-IN-4
GENERAL CATALOGUE

DXR-IN-4

HY-170783 · 50 mg

MedChemExpress · Cat: HY-170783

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medchemexpress.com/dxr-in-4.html
Catalog No: HY-170783
Category: Anti-infection
Pack Size: 50 mg
Brand: MedChemExpress

Description

DXR-IN-4 Compound 12a is the inhibitor for 1-deoxy-D-xylulose 5-phosphate reductoisomerase DXR . DXR-IN-4 inhibits DXR in Plasmodium falciparum Pf DXR, Escherichia coli Ec DXR, and Mycobacterium tuberculosis Mt DXR with IC50s of 18, 4.9 and 89 nM, respectively. DXR-IN-4 exhibits antimalarial activity that inhibits P. falciparum strains 3D7 and Dd2 with IC50 of 11 ?M and 12 ?M.

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