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EGFR/ErbB-2/ErbB-4 inhibitor-3
GENERAL CATALOGUE

EGFR/ErbB-2/ErbB-4 inhibitor-3

HY-103440 · 5 mg

MedChemExpress · Cat: HY-103440

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Catalog No: HY-103440
CAS No: 881001-19-0
Category: JAK STAT Signaling
Pack Size: 5 mg
Brand: MedChemExpress

Description

EGFR/ErbB-2/ErbB-4 inhibitor-3 compound 29 is a potent tyrosine kinase inhibitor with IC50s of 0.3, 1.1, 0.5, 2.5, 24 nM for erbB1, erbB2, erbB4, EGF, HER, respectively. EGFR/ErbB-2/ErbB-4 inhibitor-3 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition CuAAc with molecules containing Azide groups.

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