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EGFR/HER2/DHFR-IN-1
GENERAL CATALOGUE

EGFR/HER2/DHFR-IN-1

HY-151154 · 50 mg

MedChemExpress · Cat: HY-151154

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Catalog No: HY-151154
CAS No: 2820126-37-0
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress

Description

EGFR/HER2/DHFR-IN-1 is a potent anticancer agent with high selectivity against MCF-7 breast cancer cells. EGFR/HER2/DHFR-IN-1 is a multiple inhibitor of EGFR/HER2 kinase and DHFR, with IC50s of 0.153 ?M, 0.108 ?M, 0.291 ?M, respectively. EGFR/HER2/DHFR-IN-1 arrests cell cycle at G1/S and induces cells apoptosis.

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