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EGFR/HER2-IN-11
GENERAL CATALOGUE

EGFR/HER2-IN-11

HY-160613 · 50 mg

MedChemExpress · Cat: HY-160613

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Catalog No: HY-160613
CAS No: 1346176-20-2
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress

Description

EGFR/HER2-IN-11 compound 20 is an orally active dual inhibitor for human epidermal growth factor receptor 2 HER2 and epidermal growth factor receptor EGFR , with IC50s of 7.7 and 22 nM, respectively. EGFR/HER2-IN-11 exhibits antitumor efficacy and inhibits proliferation against cancer cells BT-474 with GI50 of 601 nM.

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