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EGFR/HER2-IN-8
GENERAL CATALOGUE

EGFR/HER2-IN-8

HY-151161 · 50 mg

MedChemExpress · Cat: HY-151161

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Catalog No: HY-151161
CAS No: 2820126-32-5
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress

Description

EGFR/HER2-IN-8 compound 34 is a EGFR/HER2 and DHFR inhibitor. EGFR/HER2-IN-8 inhibits EGFR kinase, HER2 kinase and DHFR with IC50s of 0.45, 0.244 and 5.669 ?M, respectively. EGFR/HER2-IN-8 shows anticancer activity against several cancer cell lines with high safety profile and selectivity indices. EGFR/HER2-IN-8 can be used for the research of cancer.

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