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EGFR-IN-132
GENERAL CATALOGUE

EGFR-IN-132

HY-169308 · 50 mg

MedChemExpress · Cat: HY-169308

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medchemexpress.com/egfr-in-132.html
Catalog No: HY-169308
CAS No: 2809982-20-3
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress

Description

EGFR-IN-132 Compound 23 is an inhibitor for EGFR, that inhibits the EGFR wildtype, L858R/T790M, d19/T790M, L858R/T790M/C797S, and d19/T790M/C797S mutans with IC50 of 1.6, 0.025, 0.019, 0.022, and 0.029 nM. EGFR-IN-132 exhibits good pharmacokinetics characteristics with high oral exposure.

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