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EGFR-IN-61
GENERAL CATALOGUE

EGFR-IN-61

HY-147860 · 50 mg

MedChemExpress · Cat: HY-147860

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Manufacturer product page

medchemexpress.com/egfr-in-61.html
Catalog No: HY-147860
CAS No: 2890261-81-9
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress

Description

EGFR-IN-61 compound 22a is a potent EGFR kinase inhibitor, with IC50 values of 42 nM L858R/T790 M , 137 nM L858R/T790 M/C797S , and 743 nM WT , respectively. EGFR-IN-61 shows antiproliferative activity against A549 and H1975 cell lines, with IC50 values of 2.14 and 1.82 ?M, respectively.

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