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EGFR-IN-90
GENERAL CATALOGUE

EGFR-IN-90

HY-156457 · 50 mg

MedChemExpress · Cat: HY-156457

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medchemexpress.com/egfr-in-90.html
Catalog No: HY-156457
CAS No: 3008611-00-2
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress

Description

EGFR-IN-90 compound 34 is an orally active EGFR inhibitor. EGFR-IN-90 shows inhibitory activity against EGFRL858R/T790M/C797S with an IC50 of 5.1 nM and inhibits the proliferation of the H1975-TM cell line harboring EGFRL858R/T790M/C797S with an IC50 of 0.05 ?M. EGFR-IN-90 and inhibits tumor growth in the H1975-TM xenograft tumor model.

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