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EGFR kinase inhibitor 1
GENERAL CATALOGUE

EGFR kinase inhibitor 1

HY-143246 · 50 mg

MedChemExpress · Cat: HY-143246

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Catalog No: HY-143246
CAS No: 2413958-04-8
Category: Apoptosis
Pack Size: 50 mg
Brand: MedChemExpress

Description

EGFR kinase inhibitor 1 is a potent EGFR inhibitor with IC50s of 37, 1.7, >300 nM for WT, l885R/T790M, L858R/T790M/C797S, respectively. EGFR kinase inhibitor 1 induces apoptosis and cell cycle arrest at G0/G1-phase. EGFR kinase inhibitor 1 inhibits the cell motility. EGFR kinase inhibitor 1 shows antiproliferative and anti-tumor activity.

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