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EGFR kinase inhibitor 3
GENERAL CATALOGUE

EGFR kinase inhibitor 3

HY-162299 · 5 mg

MedChemExpress · Cat: HY-162299

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Catalog No: HY-162299
CAS No: 2922402-03-5
Category: JAK STAT Signaling
Pack Size: 5 mg
Brand: MedChemExpress

Description

EGFR kinase inhibitor 3 compound 2 is a bivalent ATP-allosteric EGFR kinase inhibitor with IC50s of <10 nM, 1.5 nM, 0.059 nM, 0.064 nM for WT EGFR, EGFR-activating mutations L858R, L858R/T790M and L858R/T790M/C797S, respectively. EGFR kinase inhibitor 3 is a C-linked inhibitor.

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