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EGFR T790M/L858R-IN-7
GENERAL CATALOGUE

EGFR T790M/L858R-IN-7

HY-158178 · 50 mg

MedChemExpress · Cat: HY-158178

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Catalog No: HY-158178
CAS No: 3032760-90-7
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress

Description

EGFR T790M/L858R-IN-7 Compound 72 is a novel pyrimidine compound that inhibits the EGFR T790M and L858R mutation with a high efficacy 93 % inhibition rate at 0.05 ?M . EGFR T790M/L858R-IN-7 functions by specifically binding to the kinase domain of EGFR, thereby inhibiting its phosphorylation activity.

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