EPI-001 (Standard)

Description

EPI-001 Standard is the analytical standard of EPI-001. This product is intended for research and analytical applications. EPI-001, a selective inhibitor of Androgen Receptor AR , targets transactivation unit 5 Tau-5 of the AR. EPI-001 can inhibit transactivation of the AR amino-terminal domain NTD , with an IC50 of 6 ?M. EPI-001 is also a selective modulator of PPAR?. EPI-001 is active against castration-resistant prostate cancer.